Can a pill that blocks multiple cancer proteins shrink Hard-to-Treat tumors?

NCT ID NCT03917043

First seen Jul 23, 2026 · Last updated Jul 24, 2026 · Updated 1 time

Summary

This early-phase trial is testing an experimental oral drug called APG-2449 in people with advanced solid tumors, including certain lung cancers, mesothelioma, esophageal cancer, and ovarian cancer. APG-2449 is designed to block several proteins (FAK, ALK, and ROS1) that help cancer cells grow. The study aims to find the safest dose and understand how the drug moves through the body.

What this could mean

Our plain-language read of the trial. This is informational only — not medical advice or a prediction.

Active substance
an experimental oral drug called APG-2449, a multi-targeted tyrosine kinase inhibitor that blocks FAK, ALK, and ROS1 proteins
What this could lead to
If it works, this could point toward a new treatment option for certain advanced solid tumors, especially lung cancers with specific gene changes.
What could go wrong
This is an early phase 1 trial, so the drug may not work as hoped or could cause unexpected side effects. The safe dose and effectiveness are still unknown.

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Conditions

The condition(s) this trial relates to.

As listed by the trial registrant

The condition terms exactly as the trial's registrant entered them.

Contacts and locations

Study contacts

  • Contact

    Phone: •••-•••-•••• Email: •••••@•••••

Locations

  • Beijing Cancer Hospital

    RECRUITING

    Beijing, Beijing Municipality, 100142, China

    Contact Email: •••••@•••••

    Contact

    Contact Email: •••••@•••••

    Contact

  • Fujian Cancer Hospital

    NOT_YET_RECRUITING

    Fuzhou, Fujian, 350014, China

    Contact

    Contact

  • Fujian Medical University Union Hospital

    NOT_YET_RECRUITING

    Fuzhou, Fujian, 350001, China

    Contact

    Contact

  • Henan Provincial Oncology Hospital

    RECRUITING

    Zhengzhou, Henan, China

    Contact

  • Hunan Provincial Oncology Hospital

    RECRUITING

    Changsha, Hunan, China

    Contact

  • Sun-Yat Sen University Cancer Center

    RECRUITING

    Guangzhou, Guangdong, 510060, China

    Contact Phone: •••-•••-•••• Email: •••••@•••••

  • The First affiliated hospital, Sun Yat-sen University

    RECRUITING

    Guangzhou, Guangdong, China

    Contact

  • Union Hospital medical college Huazhong University of Science and Technology

    RECRUITING

    Wuhan, Hubei, China

    Contact

  • Zhejiang Provincial Oncology Hospital

    RECRUITING

    Hangzhou, Zhejiang, China

    Contact

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